TargetMol

Enciprazine

Product Code:
 
TAR-T27262
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T27262-5mg5mg£850.00
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TAR-T27262-50mg50mg£1,661.00
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Quantity:
TAR-T27262-100mg100mg£2,079.00
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Further Information

Bioactivity:
Enciprazine, a GABA receptor agonist, is used potentially for the treatment of anxiety disorders.
CAS:
68576-86-3
Formula:
C23H32N2O6
Molecular Weight:
432.517
Purity:
0.98
SMILES:
COc1ccccc1N1CCN(CC(O)COc2cc(OC)c(OC)c(OC)c2)CC1

References

1. Matheson GK, Knowles A, Gage D, Michel C, Guthrie D, Bauer C, Blackbourne J, Weinzapfel D. Modification of hypothalamic-pituitary-adrenocortical activity by serotonergic agents in the rat. Pharmacology. 1997 Aug;55(2):59-65. PubMed PMID: 9323305. 2. Scatina JA, Lockhead SR, Cayen MN, Sisenwine SF. Metabolic disposition of enciprazine, a non-benzodiazepine anxiolytic drug, in rat, dog and man. Xenobiotica. 1991 Dec;21(12):1591-604. PubMed PMID: 1686125. 3. Engel J, Fleischhauer I, Jakovlev V, Kleemann A, Kutscher B, Nickel B, Rauer H, Werner U, Szelenyi I, Johanson CE, et al. Chemistry and pharmacology of the non-benzodiazepine anxiolytic enciprazine and related compounds. J Med Chem. 1990 Nov;33(11):2976-81. PubMed PMID: 1977910. 4. Scheibe G, Grohmann R, Buchheim P. Pilot study on the therapeutic efficacy, clinical safety, and dosage finding of enciprazine in out-patients with anxious and anxious-depressive syndromes. Arzneimittelforschung. 1990 Jun;40(6):644-6. PubMed PMID: 2204343.