TargetMol

FR-217840

Product Code:
 
TAR-T27382
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T27382-5mg5mg£1,171.00
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TAR-T27382-50mg50mg£2,303.00
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Quantity:
TAR-T27382-100mg100mg£3,042.00
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Further Information

Bioactivity:
FR-217840, a novel matrix metalloproteinase inhibitor, successfully suppresses joint destruction and suggest that FR217840 may have potential as a novel anti-rheumatic drug.
CAS:
848444-16-6
Formula:
C16H18FN3O6S3
Molecular Weight:
463.51
Purity:
0.98
SMILES:
CS(=O)(=O)N1CCN([C@@H](C1)C(=O)NO)S(=O)(=O)c1ccc(s1)-c1ccc(F)cc1

References

1. Ishikawa T, Nishigaki F, Miyata S, Hirayama Y, Minoura K, Imanishi J, Neya M, Mizutani T, Imamura Y, Ohkubo Y, Mutoh S. Prevention of progressive joint destruction in adjuvant induced arthritis in rats by a novel matrix metalloproteinase inhibitor, FR217840. Eur J Pharmacol. 2005 Jan 31;508(1-3):239-47. Epub 2005 Jan 12. Erratum in: Eur J Pharmacol. 2005 May 16;515(1-3):188. PubMed PMID: 15680277.