TargetMol

GR 128107

Product Code:
 
TAR-T27429
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T27429-5mg5mg£850.00
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TAR-T27429-50mg50mg£1,661.00
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Quantity:
TAR-T27429-100mg100mg£2,079.00
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Further Information

Bioactivity:
GR 128107 is an antagonist of melatonin receptor.
CAS:
190328-44-0
Formula:
C16H20N2O2
Molecular Weight:
272.348
Purity:
0.98
SMILES:
COc1ccc2[nH]cc(C3CCCN(C3)C(C)=O)c2c1

References

1. Crespi F. Influence of melatonin or its antagonism on alcohol consumption in ethanol drinking rats: a behavioral and in vivo voltammetric study. Brain Res. 2012 May 3;1452:39-46. doi: 10.1016/j.brainres.2011.10.050. PubMed PMID: 22464879. 2. Teh MT, Sugden D. The putative melatonin receptor antagonist GR128107 is a partial agonist on Xenopus laevis melanophores. Br J Pharmacol. 1999 Mar;126(5):1237-45. PubMed PMID: 10205014; PubMed Central PMCID: PMC1565880.