TargetMol

GRI918013

Product Code:
 
TAR-T27433
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T27433-5mg5mg£850.00
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TAR-T27433-50mg50mg£1,661.00
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Quantity:
TAR-T27433-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
GRI918013 is an ATX inhibitor.
CAS:
313685-55-1
Formula:
C17H15Cl2FN2O4S
Molecular Weight:
433.28
Purity:
0.98
SMILES:
Fc1cccc(NC(=O)c2cc(c(Cl)cc2Cl)S(=O)(=O)N2CCOCC2)c1

References

1. Fells, James I.; Lee, Sue Chin; Norman, Derek D.; Tsukahara, Ryoko; Kirby, Jason R.; Nelson, Sandra; Seibel, William; Papoian, Ruben; Patil, Renukadevi; Miller, Duane D.; et al. Targeting the hydrophobic pocket of autotaxin with virtual screening of inhibitors identifies a common aromatic sulfonamide structural motif. FEBS Journal (2014), 281(4), 1017-1028. 2. Fells, James I.; Lee, Sue Chin; Fujiwara, Yuko; Norman, Derek D.; Lim, Keng Gat; Tsukahara, Ryoko; Liu, Jianxiong; Patil, Renukadevi; Miller, Duane D.; Kirby, R. Jason; et al. Hits of a high-?throughput screen identify the hydrophobic pocket of autotaxin?/lysophospholipase D as an inhibitory surface. Molecular Pharmacology (2013), 84(3), 415-424.