TargetMol

GSK 1440115

Product Code:
 
TAR-T27441
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T27441-5mg5mg£1,010.00
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Quantity:
TAR-T27441-50mg50mg£1,982.00
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Quantity:
TAR-T27441-100mg100mg£2,560.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
GSK 1440115, an orally active urotensin II receptor antagonist, is used to treat asthma.
CAS:
1003878-16-7
Formula:
C30H29Cl2N3O6
Molecular Weight:
598.48
Purity:
0.98
SMILES:
CN([C@@H](CN1CCOCC1)c1ccc(cc1)-c1ccc(cc1)C(O)=O)C(=O)CN1C(=O)COc2cc(Cl)c(Cl)cc12

References

1. Behm DJ, Aiyar NV, Olzinski AR, McAtee JJ, Hilfiker MA, Dodson JW, Dowdell SE, Wang GZ, Goodman KB, Sehon CA, Harpel MR, Willette RN, Neeb MJ, Leach CA, Douglas SA. GSK1562590, a slowly dissociating urotensin-II receptor antagonist, exhibits prolonged pharmacodynamic activity ex vivo. Br J Pharmacol. 2010 Sep;161(1):207-28. doi: 10.1111/j.1476-5381.2010.00889.x. PubMed PMID: 20718751; PubMed Central PMCID: PMC2962828.