TargetMol

GSK1614343

Product Code:
 
TAR-T27451
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T27451-5mg5mg£410.00
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Quantity:
TAR-T27451-50mg50mg£1,661.00
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Quantity:
TAR-T27451-100mg100mg£2,079.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
GSK1614343 is an antagonist of ghrelin receptor.
CAS:
1092476-84-0
Formula:
C22H23F6N5O
Molecular Weight:
487.45
Purity:
0.98
SMILES:
[H][C@]12CCCN1CCN(C2)[C@@H](C(=O)NNc1cc(cc(c1)C(F)(F)F)C(F)(F)F)c1cccnc1

References

1. Costantini VJ, Vicentini E, Sabbatini FM, Valerio E, Lepore S, Tessari M, Sartori M, Michielin F, Melotto S, Bifone A, Pich EM, Corsi M. GSK1614343, a novel ghrelin receptor antagonist, produces an unexpected increase of food intake and body weight in rodents and dogs. Neuroendocrinology. 2011;94(2):158-68. doi: 10.1159/000328968. Erratum in: Neuroendocrinology. 2012;95(3):247. Bifone, Angelo [added]. PubMed PMID: 21778696.