TargetMol

GSK931145

Product Code:
 
TAR-T27494
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T27494-5mg5mg£850.00
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TAR-T27494-50mg50mg£1,661.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T27494-100mg100mg£2,079.00
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This product comes from: United States.
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  • Further Information
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Further Information

Bioactivity:
GSK931145 is a positron emission tomography (PET) radioligand, it is suitable for quantifying glycine transporter (GlyT1) availability in the living brain.
CAS:
896117-64-9
Formula:
C23H30N2O
Molecular Weight:
350.506
Purity:
0.98
SMILES:
CN(C)C1(CCCC1)[C@@H](NC(=O)c1c(C)cccc1C)c1ccccc1

References

1. Zheng MQ, Lin SF, Holden D, Naganawa M, Ropchan JR, Najafzaden S, Kapinos M, Tabriz M, Carson RE, Hamill TG, Huang Y. Comparative evaluation of two glycine transporter 1 radiotracers [11C]GSK931145 and [18F]MK-6577 in baboons. Synapse. 2016 Mar;70(3):112-20. doi: 10.1002/syn.21879. PubMed PMID: 26671330. 2. Chopra A. (11)C-Labeled GSK931145. 2012 Mar 2 [updated 2012 Apr 19]. Molecular Imaging and Contrast Agent Database (MICAD) [Internet]. Bethesda (MD): National Center for Biotechnology Information (US); 2004-2013. Available from http://www.ncbi.nlm.nih.gov/books/NBK92277/ PubMed PMID: 22536614. 3. Gunn RN, Murthy V, Catafau AM, Searle G, Bullich S, Slifstein M, Ouellet D, Zamuner S, Herance R, Salinas C, Pardo-Lozano R, Rabiner EA, Farre M, Laruelle M. Translational characterization of [11C]GSK931145, a PET ligand for the glycine transporter type 1. Synapse. 2011 Dec;65(12):1319-32. doi: 10.1002/syn.20966. PubMed PMID: 21688322. 4. Bullich S, Slifstein M, Passchier J, Murthy NV, Kegeles LS, Kim JH, Xu X, Gunn RN, Herance R, Gispert JD, Guti?rrez A, Farr? M, Laruelle M, Catafau AM. Biodistribution and radiation dosimetry of the glycine transporter-1 ligand 11C-GSK931145 determined from primate and human whole-body PET. Mol Imaging Biol. 2011 Aug;13(4):776-84. doi: 10.1007/s11307-010-0398-6. PubMed PMID: 20730499.