TargetMol

JNJ-20788560

Product Code:
 
TAR-T27667
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T27667-1mg1mg£352.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T27667-1mL1 mL * 10 mM (in DMSO)£542.00
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Quantity:
TAR-T27667-5mg5mg£736.00
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Quantity:
TAR-T27667-10mg10mg£978.00
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Quantity:
TAR-T27667-25mg25mg£1,348.00
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Quantity:
TAR-T27667-50mg50mg£1,661.00
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Quantity:
TAR-T27667-100mg100mg£2,079.00
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Quantity:
TAR-T27667-500mg500mg£4,006.00
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Quantity:
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This product comes from: United States.
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  • Further Information
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Further Information

Bioactivity:
JNJ-20788560 is a delta opioid receptor (DOR) agonist analgesics. It is selective for DOR over the mu opioid receptor (MOR).
CAS:
825649-28-3
Formula:
C25H28N2O2
Molecular Weight:
388.511
Pathway:
Endocrinology/Hormones|GPCR/G Protein|Neuroscience
Purity:
0.98
SMILES:
CCN(CC)C(=O)c1ccc2C(=C3CC4CCC(C3)N4)c3ccccc3Oc2c1
Target:
Opioid Receptor

References

1. Codd EE, Ma J, Zhang SP, Stone DJ Jr, Colburn RW, Brandt MR, Chevalier KM, Zhu Y, Peng S, Cai C, Acton PD, Flores CM. Ex vivo delta opioid receptor autoradiography: CNS receptor occupancy of two novel compounds over their antihyperalgesic dose range. Pharmacol Biochem Behav. 2010 Aug;96(2):130-5. doi: 10.1016/j.pbb.2010.04.020. Epub 2010 May 12. PubMed PMID: 20438745. 2. Codd EE, Carson JR, Colburn RW, Stone DJ, Van Besien CR, Zhang SP, Wade PR, Gallantine EL, Meert TF, Molino L, Pullan S, Razler CM, Dax SL, Flores CM. JNJ-20788560 [9-(8-azabicyclo[3.2.1]oct-3-ylidene)-9H-xanthene-3-carboxylic acid diethylamide], a selective delta opioid receptor agonist, is a potent and efficacious antihyperalgesic agent that does not produce respiratory depression, pharmacologic tolerance, or physical dependence. J Pharmacol Exp Ther. 2009 Apr;329(1):241-51. doi: 10.1124/jpet.108.146969. Epub 2009 Jan 16. PubMed PMID: 19151246.