TargetMol

JNJ-54166060

Product Code:
 
TAR-T27688
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T27688-5mg5mg£850.00
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Quantity:
TAR-T27688-50mg50mg£1,661.00
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Quantity:
TAR-T27688-100mg100mg£2,079.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
JNJ-54166060 is a potent P2X7 antagonist. rP2X7 IC50=4 nM; rP2X7 IC50=115nM; HLM/RLM = 0.35/0.64, ED50 = 2.3 mg/kg in rats. JNJ-54166060 possesses a unique CYP profile and was found to be a regioselective inhibitor of midazolam CYP3A metabolism.
CAS:
1627900-42-8
Formula:
C20H15ClF4N4O
Molecular Weight:
438.81
Purity:
0.98
SMILES:
C[C@H]1N(CCc2c1ncn2-c1ccc(F)cn1)C(=O)c1cccc(c1Cl)C(F)(F)F