TargetMol

MRS1097

Product Code:
 
TAR-T28098
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T28098-5mg5mg£850.00
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TAR-T28098-50mg50mg£1,661.00
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Quantity:
TAR-T28098-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
MRS1097 is a selective antagonist A3 adenosine receptor.
CAS:
185259-16-9
Formula:
C26H27NO4
Molecular Weight:
417.505
Purity:
0.98
SMILES:
CCOC(=O)C1=C(C)NC(=C(C1C=Cc1ccccc1)C(=O)OCC)c1ccccc1

References

1. Durand IH, Green RD. Cloning of a chick A3 adenosine receptor: characterization of ligand binding and receptor-effector coupling of chick A1 and A3 adenosine receptors. Naunyn Schmiedebergs Arch Pharmacol. 2001 Jan;363(1):81-6. PubMed PMID: 11191840. 2. Mitchell CH, Peterson-Yantorno K, Carr? DA, McGlinn AM, Coca-Prados M, Stone RA, Civan MM. A3 adenosine receptors regulate Cl- channels of nonpigmented ciliary epithelial cells. Am J Physiol. 1999 Mar;276(3 Pt 1):C659-66. PubMed PMID: 10069993. 3. Jacobson KA, Park KS, Jiang JL, Kim YC, Olah ME, Stiles GL, Ji XD. Pharmacological characterization of novel A3 adenosine receptor-selective antagonists. Neuropharmacology. 1997 Sep;36(9):1157-65. PubMed PMID: 9364471; PubMed Central PMCID: PMC3433714. 4. Jiang J, van Rhee AM, Chang L, Patchornik A, Ji XD, Evans P, Melman N, Jacobson KA. Structure-activity relationships of 4-(phenylethynyl)-6-phenyl-1,4-dihydropyridines as highly selective A3 adenosine receptor antagonists. J Med Chem. 1997 Aug 1;40(16):2596-608. PubMed PMID: 9258367.