Oxendolone

Product Code:

TAR-T28280

Product Group:

Inhibitors and Activators

Supplier:

TargetMol

Regulatory Status:

RUO

Shipping:

cool pack

Storage:

-20℃

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Code	Size	Price

TAR-T28280-5mg

5mg

£850.00

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Quantity:

Prices exclude any Taxes / VAT

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Further Information

Bioactivity:

Oxendolone is a steroidal progestin and antiandrogen. Oxendolone binds to the progesterone receptor (Ki = 20 nM) and androgen receptor (AR) (Ki = 320 nM) and acts as a weak but clinically relevant inhibitor of 5α-reductase.

CAS:

33765-68-3

Formula:

C20H30O2

Molecular Weight:

302.458

Purity:

0.98

SMILES:

CC[C@H]1C[C@H]2[C@@H]3CCC4=CC(=O)CC[C@@H]4[C@H]3CC[C@]2(C)[C@H]1O

Documents

References

1. Hikichi Y, Yamaoka M, Kusaka M, Hara T. Selective androgen receptor modulator activity of a steroidal antiandrogen TSAA-291 and its cofactor recruitment profile. Eur J Pharmacol. 2015 Oct 15;765:322-31. doi: 10.1016/j.ejphar.2015.08.052. Epub 2015 Sep 1. PubMed PMID: 26335395. 2. Matsuda H, Yamazaki M, Naruo S, Asanuma Y, Kubo M. Anti-androgenic and hair growth promoting activities of Lygodii spora (spore of Lygodium japonicum) I. Active constituents inhibiting testosterone 5alpha-reductase. Biol Pharm Bull. 2002 May;25(5):622-6. PubMed PMID: 12033503. 3. Yamada K, Komatsu H, Ohta A. Effects of 3,6-dimethylpyrazine-2-thiol on reproductive and accessory reproductive organs in male rats. Biol Pharm Bull. 1996 Mar;19(3):360-3. PubMed PMID: 8924900. 4. Iguchi H, Ikeuchi T, Kai Y, Yoshida H. [Influence of anti-androgen therapy for prostatic hypertrophy on lipid metabolism]. Hinyokika Kiyo. 1994 Mar;40(3):215-9. Japanese. PubMed PMID: 7513937.