TargetMol

PD 122860

Product Code:
 
TAR-T28321
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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TAR-T28321-5mg5mg£850.00
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TAR-T28321-50mg50mg£1,661.00
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TAR-T28321-100mg100mg£2,079.00
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Further Information

Bioactivity:
PD 122860 is a dihydropyridine with calcium channel blocking and sodium channel stimulating properties. In the rat heart, PD 122860 increased left ventricular contractility, decreased coronary resistance and altered the shape of the electrocardiogram T-wave. PD 122860 selectively relaxed potassium-contracted aortic rings and inhibited [3H]nitrendipine binding to rat brain membranes.
CAS:
122576-86-7
Formula:
C23H20F3N3O4S
Molecular Weight:
491.49
Purity:
0.98
SMILES:
CCOC(=O)C1=C(CS(=O)(=O)c2ccncc2)NC(C)=C(C#N)C1c1ccccc1C(F)(F)F

References

1. Haleen SJ, Steffen RP, Sircar I, Major TC, Taylor MD, Pugsley TA, Weishaar RE. PD 122860: a novel dihydropyridine with sodium channel stimulating and calcium channel blocking properties. J Pharmacol Exp Ther. 1989 Jul;250(1):22-30. PubMed PMID: 2473188.