TargetMol

PI3KD/V-IN-01

Product Code:
 
TAR-T28413
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T28413-5mg5mg£850.00
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Quantity:
TAR-T28413-50mg50mg£1,661.00
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Quantity:
TAR-T28413-100mg100mg£2,079.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
PI3KD/V-IN-01 is a potent ATP-competitive PI3Kδ/Vps34 dual inhibitor.
CAS:
1807551-44-5
Formula:
C21H25Cl2N5O3S2
Molecular Weight:
530.48
Purity:
0.98
SMILES:
Cl.Cc1nc(NC(=O)CN)sc1-c1cnc(Cl)c(NS(=O)(=O)c2ccc(cc2)C(C)(C)C)c1

References

1. Liu X, Wang A, Liang X, Liu J, Zou F, Chen C, Zhao Z, Deng Y, Wu H, Qi Z, Wang B, Wang L, Liu F, Xu Y, Wang W, Fernandes SM, Stone RM, Galinsky IA, Brown JR, Loh T, Griffin JD, Zhang S, Weisberg EL, Zhang X, Liu J, Liu Q. Simultaneous inhibition of Vps34 kinase would enhance PI3K? inhibitor cytotoxicity in the B-cell malignancies. Oncotarget. 2016 Aug 16;7(33):53515-53525. doi: 10.18632/oncotarget.10650. PubMed PMID: 27447747; PubMed Central PMCID: PMC5288202.