TargetMol

RN9893 HCl

Product Code:
 
TAR-T28548
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T28548-5mg5mg£850.00
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Quantity:
TAR-T28548-50mg50mg£1,661.00
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Quantity:
TAR-T28548-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
RN9893 HCl is a selective TRPV4 receptor antagonist, it inhibits human, rat and murine variants of TRPV4.
CAS:
1803003-68-0
Formula:
C21H24ClF3N4O5S
Molecular Weight:
536.95
Purity:
0.98
SMILES:
Cl.CC(C)N1CCN(CC1)S(=O)(=O)c1ccc(NC(=O)c2ccc(cc2[N+]([O-])=O)C(F)(F)F)cc1

References

1. Wei ZL, Nguyen MT, O'Mahony DJ, Acevedo A, Zipfel S, Zhang Q, Liu L, Dourado M, Chi C, Yip V, DeFalco J, Gustafson A, Emerling DE, Kelly MG, Kincaid J, Vincent F, Duncton MA. Identification of orally-bioavailable antagonists of the TRPV4 ion-channel. Bioorg Med Chem Lett. 2015 Sep 15;25(18):4011-5. doi: 10.1016/j.bmcl.2015.06.098. Epub 2015 Jul 6. PubMed PMID: 26235950.