TargetMol

RTI-371

Product Code:
 
TAR-T28620
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T28620-5mg5mg£1,010.00
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TAR-T28620-50mg50mg£1,982.00
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Quantity:
TAR-T28620-100mg100mg£2,560.00
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This product comes from: United States.
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Further Information

Bioactivity:
RTI-371 is a potent and selective dopamine reuptake inhibitor in vitro.
CAS:
652978-45-5
Formula:
C24H25ClN2O
Molecular Weight:
392.93
Purity:
0.98
SMILES:
[H][C@@]12CC[C@@]([H])([C@H]([C@H](C1)c1ccc(C)cc1)c1cc(no1)-c1ccc(Cl)cc1)N2C

References

1. Navarro HA, Howard JL, Pollard GT, Carroll FI. Positive allosteric modulation of the human cannabinoid (CB) receptor by RTI-371, a selective inhibitor of the dopamine transporter. Br J Pharmacol. 2009 Apr;156(7):1178-84. doi: 10.1111/j.1476-5381.2009.00124.x. PubMed PMID: 19226282; PubMed Central PMCID: PMC2697692. 2. Hiranita T, Wilkinson DS, Hong WC, Zou MF, Kopajtic TA, Soto PL, Lupica CR, Newman AH, Katz JL. 2-isoxazol-3-phenyltropane derivatives of cocaine: molecular and atypical system effects at the dopamine transporter. J Pharmacol Exp Ther. 2014 May;349(2):297-309. doi: 10.1124/jpet.113.212738. Erratum in: J Pharmacol Exp Ther. 2014 Jun 1;349(3):534. PubMed PMID: 24518035; PubMed Central PMCID: PMC3989806. 3. Carroll FI, Pawlush N, Kuhar MJ, Pollard GT, Howard JL. Synthesis, monoamine transporter binding properties, and behavioral pharmacology of a series of 3beta-(substituted phenyl)-2beta-(3'-substituted isoxazol-5-yl)tropanes. J Med Chem. 2004 Jan 15;47(2):296-302. PubMed PMID: 14711303.