TargetMol

SDZ-216525

Product Code:
 
TAR-T28738
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T28738-5mg5mg£1,091.00
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Quantity:
TAR-T28738-50mg50mg£2,143.00
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Quantity:
TAR-T28738-100mg100mg£2,801.00
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Further Information

Bioactivity:
SDZ-216525, a 5-HT1A receptor antagonist, inhibits the tracheal contractions induced both by NKA (10 nM-3 microM) and 5-HT (10 nM-10 microM) (n=4-10).
CAS:
141533-35-9
Formula:
C25H28N4O5S
Molecular Weight:
496.58
Purity:
0.98
SMILES:
COC(=O)c1cc2c(cccc2[nH]1)N1CCN(CCCCN2C(=O)c3ccccc3S2(=O)=O)CC1

References

1. Germonpr? PR, Joos GF, Pauwels RA. Modulation by 5-HT1A receptors of the 5-HT2 receptor-mediated tachykinin-induced contraction of the rat trachea in vitro. Br J Pharmacol. 1998 Apr;123(8):1571-8. PubMed PMID: 9605563; PubMed Central PMCID: PMC1565327.