TargetMol

SM-130686

Product Code:
 
TAR-T28812
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T28812-5mg5mg£930.00
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TAR-T28812-50mg50mg£1,821.00
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Quantity:
TAR-T28812-100mg100mg£2,319.00
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Further Information

Bioactivity:
SM-130,686 is a potent, orally-active agonist of the ghrelin/growth hormone secretagogue receptor (GHSR) and growth hormone secretagogue. It has around half the potency of the endogenous agonist ghrelin as a stimulator of growth hormone release.
CAS:
259667-25-9
Formula:
C22H23ClF3N3O3
Molecular Weight:
469.89
Purity:
0.98
SMILES:
CCN(CC)CCN1C(=O)[C@@](O)(c2c1cc(cc2C(F)(F)F)C(N)=O)c1ccccc1Cl

References

1. Tokunaga T, Hume WE, Nagamine J, Kawamura T, Taiji M, Nagata R. Structure-activity relationships of the oxindole growth hormone secretagogues. Bioorganic and Medicinal Chemistry Letters. 2005 Apr 1;15(7):1789-92. PMID 15780607 2. Nagamine J, Nagata R, Seki H, Nomura-Akimaru N, Ueki Y, Kumagai K, Taiji M, Noguchi H. Pharmacological profile of a new orally active growth hormone secretagogue, SM-130686. Journal of Endocrinology. 2001 Dec;171(3):481-9. PMID 11739014