TargetMol

Telenzepine

Product Code:
 
TAR-T28941
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T28941-5mg5mg£850.00
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Quantity:
TAR-T28941-50mg50mg£1,661.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T28941-100mg100mg£2,079.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
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This product comes from: United States.
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Further Information

Bioactivity:
Telenzepine is a potent and selective M1 antimuscarinic.
CAS:
80880-90-6
Formula:
C19H23N4O2S
Molecular Weight:
371.48
Purity:
0.98
SMILES:
CN1CCN(CC(=O)C2=NC3=C(CCC=C3)[N](=O)c3csc(C)c23)CC1

References

1. Pelosi A, Menardy F, Popa D, Girault JA, Herv? D. Heterozygous Gnal mice are a novel animal model to study dystonia pathophysiology. J Neurosci. 2017 May 25. pii: 1529-16. doi: 10.1523/JNEUROSCI.1529-16.2017. [Epub ahead of print] PubMed PMID: 28546310. 2. Joseph L, Thomsen M. Effects of muscarinic receptor antagonists on cocaine discrimination in wild-type mice and in muscarinic receptor M(1), M(2), and M(4) receptor knockout mice. Behav Brain Res. 2017 Apr 22;329:75-83. doi: 10.1016/j.bbr.2017.04.023. [Epub ahead of print] PubMed PMID: 28442355. 3. Ztaou S, Maurice N, Camon J, Guiraudie-Capraz G, Kerkerian-Le Goff L, Beurrier C, Liberge M, Amalric M. Involvement of Striatal Cholinergic Interneurons and M1 and M4 Muscarinic Receptors in Motor Symptoms of Parkinson's Disease. J Neurosci. 2016 Aug 31;36(35):9161-72. doi: 10.1523/JNEUROSCI.0873-16.2016. PubMed PMID: 27581457. 4. Pediani JD, Ward RJ, Godin AG, Marsango S, Milligan G. Dynamic Regulation of Quaternary Organization of the M1 Muscarinic Receptor by Subtype-selective Antagonist Drugs. J Biol Chem. 2016 Jun 17;291(25):13132-46. doi: 10.1074/jbc.M115.712562. Epub 2016 Apr 14. PubMed PMID: 27080256; PubMed Central PMCID: PMC4933229.