TargetMol

VAL-201

Product Code:
 
TAR-T29088
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T29088-5mg5mg£850.00
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Further Information

Bioactivity:
VAL-201, an androgen receptor antagonist, is used potentially for the treatment of prostate cancer.
CAS:
957791-38-7
Formula:
C55H87N19O11
Molecular Weight:
1190.423
Purity:
0.98
SMILES:
CC[C@H](C)[C@H](NC(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](C)NC(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H]1CCCN1C(=O)[C@H](Cc1c[nH]cn1)NC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(C)=O)C(=O)N[C@@H](CCCCN)C(N)=O

References

1. Xiang DF, Xu C, Kumaran D, Brown AC, Sauder JM, Burley SK, Swaminathan S, Raushel FM. Functional annotation of two new carboxypeptidases from the amidohydrolase superfamily of enzymes. Biochemistry. 2009 Jun 2;48(21):4567-76. doi: 10.1021/bi900453u. PubMed PMID: 19358546; PubMed Central PMCID: PMC2748308. 2. Thompson AJ, Padgett CL, Lummis SC. Mutagenesis and molecular modeling reveal the importance of the 5-HT3 receptor F-loop. J Biol Chem. 2006 Jun 16;281(24):16576-82. PubMed PMID: 16595668. 3. Matsui I, Matsui E, Sakai Y, Kikuchi H, Kawarabayasi Y, Ura H, Kawaguchi S, Kuramitsu S, Harata K. The molecular structure of hyperthermostable aromatic aminotransferase with novel substrate specificity from Pyrococcus horikoshii. J Biol Chem. 2000 Feb 18;275(7):4871-9. PubMed PMID: 10671523.