TargetMol

VPC-13163

Product Code:
 
TAR-T29110
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T29110-1mg1mg£181.00
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Quantity:
TAR-T29110-1mL1 mL * 10 mM (in DMSO)£307.00
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Quantity:
TAR-T29110-5mg5mg£340.00
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Quantity:
TAR-T29110-10mg10mg£470.00
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Quantity:
TAR-T29110-25mg25mg£707.00
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Quantity:
TAR-T29110-50mg50mg£978.00
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Quantity:
TAR-T29110-100mg100mg£1,291.00
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Quantity:
TAR-T29110-500mg500mg£2,456.00
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Quantity:
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Further Information

Bioactivity:
VPC-13163 has strong anti-proliferative activity against LNCaP and Enzalutamide-resistant prostate cancer cell lines (MR49F) whereas it did not affect the growth of AR independent PC3 cell line. It also inhibits Prostate Specific Antigen (PSA) in both LNCaP and MR49F and reduces expression of AR target genes, PSA and TMPRSS2. These findings suggest that VPC-13566 exhibits AR BF3 specific mechanism of action.
CAS:
6637-10-1
Formula:
C16H14N2
Molecular Weight:
234.302
Purity:
0.985
SMILES:
C1C(Nc2ccccc12)c1c[nH]c2ccccc12

References

1. Frederick Glenn WEST, et al. Treatment of infectious disease.WO2019183729A1