TargetMol

VU0152099

Product Code:
 
TAR-T29123
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T29123-5mg5mg£108.00
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Quantity:
TAR-T29123-1mL1 mL * 10 mM (in DMSO)£130.00
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Quantity:
TAR-T29123-10mg10mg£135.00
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Quantity:
TAR-T29123-25mg25mg£209.00
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Quantity:
TAR-T29123-50mg50mg£294.00
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Quantity:
TAR-T29123-100mg100mg£431.00
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Quantity:
TAR-T29123-500mg500mg£863.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ? 93 nM).
CAS:
612514-42-8
Formula:
C18H17N3O3S
Molecular Weight:
355.41
Pathway:
Neuroscience
Purity:
0.98
SMILES:
Cc1cc(C)c2c(N)c(sc2n1)C(=O)NCc1ccc2OCOc2c1
Target:
AChR

References

1. Brady A E , Jones C K , Bridges T M , et al. Centrally Active Allosteric Potentiators of the M4 Muscarinic Acetylcholine Receptor Reverse Amphetamine-Induced Hyperlocomotor Activity in Rats[J]. Journal of Pharmacology & Experimental Therapeutics, 2008, 327(3):941-953.