TargetMol

CL 277082

Product Code:
 
TAR-T30961
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

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CodeSizePrice
TAR-T30961-5mg5mg£850.00
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This product comes from: United States.
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Further Information

Bioactivity:
CL 277082 is a boichemical.
CAS:
96224-26-9
Formula:
C26H36F2N2O
Molecular Weight:
430.584
Purity:
0.98
SMILES:
CCCCCCCN(Cc1ccc(CC(C)(C)C)cc1)C(=O)Nc1ccc(F)cc1F

References

1. Pal S, Allister E, Thomson A, Mamo JC. Cholesterol esters regulate apoB48 secretion in CaCo2 cells. Atherosclerosis. 2002 Mar;161(1):55-63. PubMed PMID: 11882317. 2. Kusunoki J, Aragane K, Kitamine T, Yamaura T, Ohnishi H. [Effect of F-1394, a potent and selective inhibitor of acyl-CoA:cholesterol acyltransferase (ACAT), on esterification of cholesterol and basolateral secretion of cholesteryl ester in Caco-2 cells]. Nihon Yakurigaku Zasshi. 1997 Dec;110(6):357-65. Japanese. PubMed PMID: 9503394. 3. Ellsworth JL, Starr JR. Inhibition of acyl coenzyme A:cholesterol acyltransferase blocks esterification but not uptake of cholesterol in Caco-2 cells. Metabolism. 1998 Mar;47(3):325-32. PubMed PMID: 9500571. 4. Hawke RL, Chapman JM, Winegar DA, Salisbury JA, Welch RM, Brown A, Franzmann KW, Sigel C. Potent hypocholesterolemic activity of novel ureido phenoxyisobutyrates correlates with their intrinsic fibrate potency and not with their ACAT inhibitory activity. J Lipid Res. 1997 Jun;38(6):1189-203. PubMed PMID: 9215547.