TargetMol

NU2058

Product Code:
 
TAR-T3186
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T3186-5mg5mg£107.00
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Quantity:
TAR-T3186-10mg10mg£136.00
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Quantity:
TAR-T3186-25mg25mg£180.00
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Quantity:
TAR-T3186-50mg50mg£240.00
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Quantity:
TAR-T3186-100mg100mg£334.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
NU2058 is a guanine-based CDK inhibitor, also inhibits DNA topoisomerase II ATPase activity.
CAS:
161058-83-9
Formula:
C12H17N5O
Molecular Weight:
247.302
Pathway:
DNA Damage/DNA Repair; Cell Cycle/Checkpoint
Purity:
0.9995
SMILES:
Nc1nc(OCC2CCCCC2)c2nc[nH]c2n1
Target:
Topoisomerase; CDK

References

1. Rigas AC, et al. Oncogene. 2007 Dec 6;26(55):7611-9. 2. Jensen LH, et al. Y Res. 2005 Aug 15;65(16):7470-7. 3. Knockaert M, et al. Trends Pharmacol Sci. 2002 Sep;23(9):417-25. 4. Arris CE, et al. J Med Chem. 2000 Jul 27;43(15):2797-804.