TargetMol

PF-CBP1 hydrochloride

Product Code:
 
TAR-T3217
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T3217-5mg5mg£102.00
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TAR-T3217-1mL1 mL * 10 mM (in DMSO)£114.00
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TAR-T3217-10mg10mg£118.00
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TAR-T3217-25mg25mg£168.00
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TAR-T3217-50mg50mg£230.00
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TAR-T3217-100mg100mg£367.00
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TAR-T3217-200mg200mg£455.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
PF-CBP1 is a highly selective inhibitor of the bromodomain of CREB-binding protein(CREBBP).It inhibits CREBBP and p300 bromodomains with IC50 of 125 and 363 nM respectively.
CAS:
2070014-93-4
Formula:
C29H37ClN4O3
Molecular Weight:
525.09
Pathway:
Chromatin/Epigenetic
Purity:
0.99
SMILES:
Cl.CCCOc1ccc(CCc2nc3cc(ccc3n2CCN2CCOCC2)-c2c(C)noc2C)cc1
Target:
Epigenetic Reader Domain; Histone Acetyltransferase

References

1. Eugene L, et al. Chem Biol. 2015, 22(12):1588-1596.