TargetMol

P 34081

Product Code:
 
TAR-T33852
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T33852-5mg5mg£850.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T33852-50mg50mg£1,661.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
TAR-T33852-100mg100mg£2,079.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
P 34081 rapidly blocks parasite cysteine proteinase activity in vivo.
CAS:
148504-23-8
Formula:
C26H33FN4O4
Molecular Weight:
484.572
Purity:
0.98
SMILES:
FCC(=O)[C@H](CCc1ccccc1)NC(=O)[C@H](Cc1ccccc1)NC(=O)NCN1CCOCC1

References

Perche O, Doly M, Ranchon-Cole I. Calpains are activated by light but their inhibition has no neuroprotective effect against light-damage. Exp Eye Res. 2009 Dec;89(6):989-94. doi: 10.1016/j.exer.2009.08.012. Epub 2009 Sep 1. PubMed PMID: 19729009. Esser RE, Angelo RA, Murphey MD, Watts LM, Thornburg LP, Palmer JT, Talhouk JW, Smith RE. Cysteine proteinase inhibitors decrease articular cartilage and bone destruction in chronic inflammatory arthritis. Arthritis Rheum. 1994 Feb;37(2):236-47. PubMed PMID: 8129779. Rosenthal PJ, Lee GK, Smith RE. Inhibition of a Plasmodium vinckei cysteine proteinase cures murine malaria. J Clin Invest. 1993 Mar;91(3):1052-6. PubMed PMID: 8450035; PubMed Central PMCID: PMC288059.