TargetMol

BPIQ-II (hydrochloride)

Product Code:
 
TAR-T36783
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T36783-5mg5mg£850.00
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Quantity:
TAR-T36783-50mg50mg£1,661.00
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Quantity:
TAR-T36783-100mg100mg£2,079.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
BPIQ-II is a linear imidazoloquinazoline that potently inhibits the tyrosine kinase activity of the epidermal growth factor receptor (EGFR; IC50 = 8 pM). It is selective for EGFR over an assortment of other tyrosine and serine/threonine kinases. Cellular studies indicate that BPIQ-II can enter cells and very selectively shut down EGF-stimulated signal transmission by binding competitively at the ATP site of EGFR.
CAS:
171179-37-6
Formula:
C15H11BrClN5
Molecular Weight:
376.64
Purity:
0.98
SMILES:
Cl.Brc1cccc(Nc2ncnc3cc4nc[nH]c4cc23)c1