TargetMol

Iralukast (CGP 45715A)

Product Code:
 
TAR-T37016
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T37016-5mg5mg£2,215.00
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TAR-T37016-50mg50mg£4,392.00
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TAR-T37016-100mg100mg£6,175.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Iralukast is a cysteinyl-leukotriene antagonist (CysLT) with a pKi of 7.8 for CysLT1.
CAS:
151581-24-7
Formula:
C38H37F3O8S
Molecular Weight:
710.76
Purity:
0.98
SMILES:
O=C(C1=CC(C2=CC=C(S[C@H]([C@H](O)C3=CC=CC(C(F)(F)F)=C3)/C=C/C=CCCCCOC4=CC=C(C(C)=O)C(O)=C4CCC)C=C2O1)=O)O

References

Magnus B?ck, et al. Update on leukotriene, lipoxin and oxoeicosanoid receptors: IUPHAR Review 7. Br J Pharmacol. 2014 Aug; 171(15): 3551-3574. Val?rie Capra, et al. Pharmacological characterization of the cysteinyl-leukotrieneantagonists CGP 45715A (iralukast) and CGP 57698 in human airways in vitro.Br J Pharmacol. 1998 Feb; 123(3): 590-598.