TargetMol

JJH260

Product Code:
 
TAR-T38107
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T38107-5mg5mg£503.00
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Quantity:
TAR-T38107-50mg50mg£2,143.00
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Quantity:
TAR-T38107-100mg100mg£2,801.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
JJH260 is an N-hydroxy hydantoin carbamate that inhibits androgen-induced gene 1 (AIG1), an enzyme that hydrolyzes fatty acid esters of hydroxy fatty acids (FAHFAs). It blocks the hydrolysis of 9-PAHSA with an IC50 value of 0.57 μM. JJH260 also inhibits the novel FAHFA hydrolase androgen-dependent TFPI-regulating protein (ADTRP; IC50 = 8.5 μM), as well as the serine hydrolase ABHD6 and the lysophospholipases LYPLA1 and LYPLA2. JJH260 inhibits the FAHFA hydrolase activity of LNCaP and T cell lysates and intact cells.
CAS:
1831135-30-8
Formula:
C29H34ClN5O5
Molecular Weight:
568.1
Purity:
0.98
SMILES:
CN(C)C(C=C1)=CC=C1C(N2CCN(C(N(OC(N3CCC(CCC4=CC=C(Cl)C=C4)CC3)=O)C5=O)=O)C5C2)=O