TargetMol

(±)-WIN 55,212 (mesylate)

Product Code:
 
TAR-T38199
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T38199-5mg5mg£105.00
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TAR-T38199-10mg10mg£139.00
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TAR-T38199-25mg25mg£237.00
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TAR-T38199-50mg50mg£369.00
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Further Information

Bioactivity:
(?)-WIN 55,212-2 is a potent aminoalkylindole cannabinoid (CB) receptor agonist with a Ki value of 62.3 and 3.3 nM for human recombinant central cannabinoid (CB1) and peripheral cannabinoid (CB2) receptors, respectively. In contrast, the enantiomer (-)-WIN 55,212-3 acts a partial inverse agonist at CB1 (pIC50 = 5.5) and as a competitive neutral antagonist of CB2, reversing the inverse agonism evoked by SR 144528 (pEC50 = 5.3). (+)-WIN 55,212 (mesylate) is a mixture of the two enantiomers, (+)-WIN 55,212-2 and (-)-WIN 55,212-3.
CAS:
137795-17-6
Formula:
C28H30N2O6S
Molecular Weight:
522.62
Purity:
0.98
SMILES:
CS(O)(=O)=O.Cc1c(C(=O)c2cccc3ccccc23)c2cccc3OCC(CN4CCOCC4)n1c23