TargetMol

TH1217

Product Code:
 
TAR-T38271
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T38271-50mg50mgEnquire
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TAR-T38271-1mg1mg£114.00
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TAR-T38271-5mg5mg£173.00
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TAR-T38271-10mg10mg£242.00
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TAR-T38271-25mg25mg£413.00
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Further Information

Bioactivity:
Potent dCTPase pyrophosphatase 1 inhibitor (IC50 = 47 nM). TH 1217 is not stable in aqueous solution. It is recommended that fresh samples are prepared and used immediately.
CAS:
1862212-48-3
Formula:
C20H17BCl2N4O6
Molecular Weight:
491.09
Purity:
0.98
SMILES:
CC1=NC2=C([N+]([O-])=O)C(Cl)=C(C=C2N1CC3=CC=C([B-]45OC(C[N+](CC(O5)=O)4C)=O)C=C3)Cl

References

Gordon DE, et, al. A SARS-CoV-2-Human Protein-Protein Interaction Map Reveals Drug Targets and Potential Drug-Repurposing. bioRxiv. 2020 Mar 22; 2020.03.22.002386. Llona-Minguez et al (2016) Discovery of the first potent and selective inhibitors of human dCTP pyrophosphatase 1. J.Med.Chem. 59 1140