TargetMol

PF-03622905

Product Code:
 
TAR-T38461
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T38461-5mg5mg£850.00
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Further Information

Bioactivity:
PF-03622905 is a potent and ATP-competitive PKC inhibitor with IC 50 s of 5.6 nM, 14.5 nM, 13 nM, 37.7 nM, and 74.1 nM for PKCα , PKCβI , PKCβII , PKCγ , and PKC? , respectively. PF-03622905 shows high specificity for PKC over other protein kinases.
CAS:
1072100-15-2
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0

References

Stephan Grant, et al. Discovery of a novel class of targeted kinase inhibitors that blocks protein kinase C signaling and ameliorates retinal vascular leakage in a diabetic rat model. Eur J Pharmacol. 2010 Feb 10;627(1-3):16-25.