TargetMol

PLX647 dihydrochloride

Product Code:
 
TAR-T39194
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T39194-5mg5mg£850.00
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This product comes from: United States.
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Further Information

Bioactivity:
PLX647 dihydrochloride is an orally active, highly specific dual FMS and KIT kinase inhibitor, with IC 50 s of 28 and 16 nM, reapectively. PLX647 dihydrochloride shows selectivity for FMS and KIT over a panel of 400 kinases at a concentration of 1 μM except FLT3 and KDR (IC 50 s=91 and 130 nM, respectively).
CAS:
1779796-38-1
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0

References

Zhang C, et al. Design and pharmacology of a highly specific dual FMS and KIT kinase inhibitor. Proc Natl Acad Sci U S A. 2013 Apr 2;110(14):5689-94.