TargetMol

CDK6/9-IN-1

Product Code:
 
TAR-T40047
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T40047-5mg5mg£850.00
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This product comes from: United States.
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Further Information

Bioactivity:
CDK6/9-IN-1 (compound 66) is an orally active active and dual CDK 6 and CDK 9 inhibitor, with IC 50 values of 40.5 nM and 39.5 nM for CDK6 anmd CDK9, respectively.
CAS:
2414373-55-8
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0

References

Yang Wang, et al. Discovery and SARs of 5-Chloro- N4-phenyl- N2-(pyridin-2-yl)pyrimidine-2,4-diamine Derivatives as Oral Available and Dual CDK 6 and 9 Inhibitors With Potent Antitumor Activity. J Med Chem. 2020 Mar 26;63(6):3327-3347.