TargetMol

Calmodulin antagonist-1

Product Code:
 
TAR-T40895
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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Further Information

Bioactivity:
Calmodulin antagonist-1 (W-7) is a calmodulin (CaM) antagonist. Calmodulin antagonist-1 inhibits calmodulin-activated Ca 2+ -phosphodiesterase (PDE) (IC 50 =28 μM). Calmodulin antagonist-1 also inhibits trypsin-treated Ca 2+ -PDE (IC 50 =375 μM) in a competitive fashion with respect to cyclic GMP and the K i value is 300 μM.
CAS:
78957-84-3
Formula:
0
Molecular Weight:
0
Purity:
0.98
SMILES:
0

References

Itoh H, et al. Direct interaction of calmodulin antagonists with Ca2+/calmodulin-dependent cyclic nucleotide phosphodiesterase. J Biochem. 1984;96(6):1721-1726.