TargetMol

CaCCinh-A01

Product Code:
 
TAR-T4330
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T4330-5mg5mg£112.00
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TAR-T4330-1mL1 mL * 10 mM (in DMSO)£116.00
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TAR-T4330-10mg10mg£138.00
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TAR-T4330-25mg25mg£222.00
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TAR-T4330-50mg50mg£322.00
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TAR-T4330-100mg100mg£495.00
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Further Information

Bioactivity:
CaCCinh-A01 is an inhibitor of the calcium-activated chloride channel (CaCC, 10 μM) and TMEM16A (IC50: 2.1 μM).
CAS:
407587-33-1
Formula:
C18H21NO4S
Molecular Weight:
347.43
Pathway:
Membrane transporter/Ion channel
Purity:
0.9992
SMILES:
CC(C)(C)C1CCc2c(C1)sc(NC(=O)c1ccco1)c2C(O)=O
Target:
Chloride channel

References

Namkung W,etal.TMEM16A inhibitors reveal TMEM16A as a minor component of calcium-activated chloridechannel conductance in airway and intestinal epithelial cells. J Biol Chem. 2011 Jan 21;286(3):2365-74. De La Fuente R, et al. Small-molecule screen identifies inhibitors of a human intestinal calcium-activated chloridechannel. Mol Pharmacol. 2008 Mar;73(3):758-68.