TargetMol

CeMMEC1

Product Code:
 
TAR-T4345
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T4345-5mg5mg£108.00
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TAR-T4345-1mL1 mL * 10 mM (in DMSO)£112.00
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TAR-T4345-10mg10mg£135.00
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TAR-T4345-25mg25mg£213.00
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TAR-T4345-50mg50mg£329.00
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TAR-T4345-100mg100mg£455.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
CeMMEC1 is an inhibitor of BRD4, and also has a great affinity for TAF1(IC50=0.9 μM).
CAS:
440662-09-9
Formula:
C19H16N2O4
Molecular Weight:
336.347
Pathway:
Chromatin/Epigenetic; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Proteases/Proteasome
Purity:
0.9926
SMILES:
Cn1cc(C(=O)Nc2ccc3OCCOc3c2)c2ccccc2c1=O
Target:
Epigenetic Reader Domain; Carboxypeptidase; DNA/RNA Synthesis

References

Sdelci S,etal. Mapping the chemical chromatin reactivation landscape identifies BRD4-TAF1 cross-talk.Nat Chem Biol. 2016 Jul;12(7):504-10.