TargetMol

TP-3654

Product Code:
 
TAR-T4523
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T4523-1mL1 mL * 10 mM (in DMSO)£112.00
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TAR-T4523-5mg5mg£112.00
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TAR-T4523-10mg10mg£132.00
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TAR-T4523-25mg25mg£193.00
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TAR-T4523-50mg50mg£269.00
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TAR-T4523-100mg100mg£368.00
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This product comes from: United States.
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Further Information

Bioactivity:
TP-3654 is a second-generation Pim kinase inhibitor (Ki values against Pim-1/3: 5/42 nM).
CAS:
1361951-15-6
Formula:
C22H25F3N4O
Molecular Weight:
418.46
Pathway:
Chromatin/Epigenetic; JAK/STAT signaling
Purity:
0.9995
SMILES:
CC(C)(O)[C@H]1CC[C@@H](CC1)Nc1ccc2ncc(-c3cccc(c3)C(F)(F)F)n2n1
Target:
Pim

References

Foulks JM, et al. A small-molecule inhibitor of PIM kinases as a potential treatment for urothelial carcinomas. Neoplasia. 2014 May;16(5):403-12.