TargetMol

Perospirone

Product Code:
 
TAR-T4576
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T4576-5mg5mg£119.00
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Quantity:
TAR-T4576-1mL1 mL * 10 mM (in DMSO)£124.00
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TAR-T4576-10mg10mg£152.00
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TAR-T4576-25mg25mg£223.00
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TAR-T4576-50mg50mg£346.00
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Quantity:
TAR-T4576-100mg100mg£542.00
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This product comes from: United States.
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Further Information

Bioactivity:
Perospirone is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors. It also displays affinity towards 5HT1A receptors as a partial agonist.
CAS:
150915-41-6
Formula:
C23H30N4O2S
Molecular Weight:
426.58
Pathway:
Neuroscience; GPCR/G Protein
Purity:
0.9945
SMILES:
[H][C@@]12CCCC[C@]1([H])C(=O)N(CCCCN1CCN(CC1)c1nsc3ccccc13)C2=O
Target:
Dopamine Receptor; 5-HT Receptor

References

Matsushita M, et al. Perospirone, a novel antipsychotic drug, inhibits marble-burying behavior via 5-HT1A receptor in mice: implications for obsessive-compulsive disorder.[J]. Journal of Pharmacological Sciences, 2005, 99(2):154-159. Ishibashi T, Ohno Y. Perospirone hydrochloride: the novel atypical antipsychotic agent with high affinities for 5-HT2, D2 and 5-HT1A receptors[J]. Biogenic Amines, 2004, 18(3):307-317. Zhou Y G, et al. Effect of the novel antipsychotic drug perospirone on P-glycoprotein function and expression in Caco-2 cells[J]. European Journal of Clinical Pharmacology, 2008, 64(7):697-703. Murata Y, et al. DNA Methylation Profiling in a Neuroblastoma Cell Line Exposed to the Antipsychotic Perospirone[J]. Pharmacopsychiatry, 2018.