TargetMol

Pipequaline hydrochloride

Product Code:
 
TAR-T4688
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T4688-1mg1mg£103.00
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TAR-T4688-5mg5mg£143.00
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TAR-T4688-10mg10mg£177.00
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TAR-T4688-25mg25mg£254.00
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TAR-T4688-50mg50mg£360.00
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TAR-T4688-100mg100mg£504.00
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This product comes from: United States.
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Further Information

Bioactivity:
Pipequaline is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It possesses a novel chemical structure that is not closely related to other drugs of this type. The drug has a similar pharmacological profile to the benzodiazepine family of drugs, but with mainly anxiolytic properties and very little sedative, amnestic or anticonvulsant effects, and so is classified as a nonbenzodiazepine anxiolytic.
CAS:
80221-58-5
Formula:
C22H25ClN2
Molecular Weight:
352.91
Pathway:
Neuroscience; Membrane transporter/Ion channel
Purity:
0.9946
SMILES:
Cl.C(Cc1cc(nc2ccccc12)-c1ccccc1)C1CCNCC1
Target:
GABA Receptor

References

Essassi D, et al. Pipequaline transport from blood to brain and liver: role of plasma protein-bound drug. J Pharm Pharmacol. 1989 Sep;41(9):595-600. Debonnel G, et al. Pipequaline acts as a partial agonist of benzodiazepine receptors: an electrophysiological study in the hippocampus of the rat. Neuropharmacology. 1987 Sep;26(9):1337-42. File SE., et al. Sedative effects of PK 9084 and PK 8165, alone and in combination with chlordiazepoxide. Br J Pharmacol. 1983 May;79(1):219-23.