TargetMol

AMZ30

Product Code:
 
TAR-T5182
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T5182-1mg1mg£96.00
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TAR-T5182-5mg5mg£127.00
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TAR-T5182-10mg10mg£157.00
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TAR-T5182-1mL1 mL * 10 mM (in DMSO)£165.00
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TAR-T5182-25mg25mg£217.00
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TAR-T5182-50mg50mg£293.00
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Quantity:
TAR-T5182-100mg100mg£400.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
AMZ30 is a selective inhibitor of PME-1 (IC50: 600 nM). It also reduces the demethylated form of PP2A in living cells.
CAS:
1313613-09-0
Formula:
C19H12FN3O6S2
Molecular Weight:
461.44
Purity:
0.9881
SMILES:
[O-][N+](=O)c1cccc(c1)S(=O)(=O)n1cccc1C=C(/C#N)S(=O)(=O)c1ccc(F)cc1

References

Bachovchin DA, et al. Discovery and optimization of sulfonyl acrylonitriles as selective, covalent inhibitors of protein phosphatase methylesterase-1. J Med Chem. 2011 Jul 28;54(14):5229-36.