TargetMol

CK1-IN-1

Product Code:
 
TAR-T5393
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T5393-1mg1mg£128.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
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TAR-T5393-5mg5mg£204.00
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TAR-T5393-1mL1 mL * 10 mM (in DMSO)£213.00
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TAR-T5393-10mg10mg£269.00
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TAR-T5393-25mg25mg£404.00
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TAR-T5393-50mg50mg£566.00
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Quantity:
TAR-T5393-100mg100mg£776.00
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This product comes from: United States.
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Further Information

Bioactivity:
CK1-IN-1, compound 1c reported in patent WO2015119579A1, is a casein kinase 1 (CK1) inhibitor. It has IC50s of 15 nM, 16 nM, 73 nM for CK1δ, and CK1ε, p38σ MAPK, respectively.
CAS:
1784751-20-7
Formula:
C24H15F2N3
Molecular Weight:
383.402
Pathway:
Metabolism; MAPK; Stem Cells
Purity:
0.9879
SMILES:
Fc1ccc(cc1)-c1nc([nH]c1-c1ccncc1)-c1ccc2ccccc2c1F
Target:
p38 MAPK; Casein Kinase

References

Filip LACO,et al. 2,4,5-tri-substituted azole-based casein kinase 1 inhibitors as inducers for cardiomyogenesis. WO2015119579A1.