TargetMol

TH-257

Product Code:
 
TAR-T7128
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7128-5mg5mg£118.00
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TAR-T7128-1mL1 mL * 10 mM (in DMSO)£124.00
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TAR-T7128-10mg10mg£145.00
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TAR-T7128-25mg25mg£221.00
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TAR-T7128-50mg50mg£331.00
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TAR-T7128-100mg100mg£491.00
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Further Information

Bioactivity:
TH 257 is a Potent and selective allosteric LIMK 1/2 inhibitor(LIMK1 and LIMK2, IC50 of 84 nM and 39 nM).
CAS:
2244678-29-1
Formula:
C24H26N2O3S
Molecular Weight:
422.54
Pathway:
Cell Cycle/Checkpoint
Purity:
0.98
SMILES:
CCCCN(Cc1ccccc1)C(=O)c1ccc(cc1)S(=O)(=O)Nc1ccccc1
Target:
LIM Kinase

References

Fabrizio M . Recent advances in the rational design and development of LIM kinase inhibitors are not enough to enter clinical trials[J]. European Journal of Medicinal Chemistry, 2018:S0223523418305075-.