TargetMol

Asperphenamate

Product Code:
 
TAR-T10390
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T10390-1mg1mg£222.00
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TAR-T10390-5mg5mg£454.00
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TAR-T10390-1mL1 mL * 10 mM (in DMSO)£494.00
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TAR-T10390-10mg10mg£603.00
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TAR-T10390-25mg25mg£863.00
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TAR-T10390-50mg50mg£1,171.00
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Quantity:
TAR-T10390-100mg100mg£1,556.00
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TAR-T10390-500mg500mg£3,058.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Asperphenamate is a fungal metabolite of Aspergillus flatiipes with anti-cancer effect (IC50s: 92.3 μM, 96.5 μM, and 97.9 μM in T47D, MDA-MB-231, and HL-60 cells).
CAS:
63631-36-7
Formula:
C32H30N2O4
Molecular Weight:
506.59
Pathway:
Others|Microbiology/Virology
Purity:
0.98
SMILES:
O=C(OC[C@@H](NC(C1=CC=CC=C1)=O)CC2=CC=CC=C2)[C@H](CC3=CC=CC=C3)NC(C4=CC=CC=C4)=O
Target:
Others|Antifungal

References

1. Alice M.Clark, et al. Synthesis of asperphenamate, a novel fungal metabolite. Phytochemistry 2. LeiYuan, et al. Total synthesis and anticancer activity studies of the stereoisomers of asperphenamate and patriscabratine. Chinese Chemical Letters Volume 21, Issue 2, February 2010, Pages 155-158. 3. Yuan L, et al. Discovery of novel cathepsin inhibitors with potent anti-metastatic effects in breast cancer cells. Bioorg Chem. 2018 Dec;81:672-680.