TargetMol

CCR2 antagonist 1

Product Code:
 
TAR-T10711
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10711-5mg5mg£524.00
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TAR-T10711-50mg50mg£2,392.00
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Quantity:
TAR-T10711-100mg100mg£3,597.00
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This product comes from: United States.
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Further Information

Bioactivity:
CCR2 antagonist 1 is a high-affinity and long-residence-time antagonist of CCR2 (Ki: 2.4 nM).
CAS:
1683534-96-4
Formula:
C28H32BrF3N2O
Molecular Weight:
549.476
Pathway:
Immunology/Inflammation; Microbiology/Virology
Purity:
0.98
SMILES:
CC(C)[C@@]1(CC[C@H](C1)N[C@@H]1CCc2cc(Br)ccc12)C(=O)N1CCc2ccc(cc2C1)C(F)(F)F
Target:
CCR

References

1. Vilums M, et al. When structure-affinity relationships meet structure-kinetics relationships: 3-((Inden-1-yl)amino)-1-isopropyl-cyclopentane-1-carboxamides as CCR2 antagonists. Eur J Med Chem. 2015 Mar 26;93:121-34.