TargetMol

CGP 20712 A

Product Code:
 
TAR-T10778
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10778-5mg5mg£370.00
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TAR-T10778-50mg50mg£1,388.00
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Quantity:
TAR-T10778-100mg100mg£2,079.00
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Further Information

Bioactivity:
CGP 20712 A (CGP 20712 mesylate) is a highly selective antagonist of β1-adrenoceptor (IC50: 0.7 nM). It shows ~10,000-fold selectivity over β2-adrenoceptors.
CAS:
105737-62-0
Formula:
C24H29F3N4O8S
Molecular Weight:
590.57
Pathway:
GPCR/G Protein; Neuroscience
Purity:
0.98
SMILES:
CS(O)(=O)=O.Cn1cc(nc1-c1ccc(OCC(O)CNCCOc2ccc(O)c(c2)C(N)=O)cc1)C(F)(F)F
Target:
Adrenergic Receptor

References

1. Dooley DJ, et al. CGP 20712 A: a useful tool for quantitating beta 1- and beta 2-adrenoceptors. Eur J Pharmacol. 1986 Oct 14;130(1-2):137-9. 2. Kitagawa Y, et al. Determination of beta-adrenoceptor subtype on rat isolated ventricular myocytes by use of highly selective beta-antagonists. Br J Pharmacol. 1995 Sep;116(1):1635-43. 3. Grino M, et al. Ontogeny of insulin-induced hypoglycemia stimulation of adrenocorticotropin secretion in the rat: role of catecholamines. Endocrinology. 1992 Dec;131(6):2763-8.