TargetMol

GDC-0927

Product Code:
 
TAR-T11380
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11380-10mg10mg£670.00
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TAR-T11380-25mg25mg£1,364.00
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Quantity:
TAR-T11380-50mg50mg£2,135.00
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This product comes from: United States.
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Further Information

Bioactivity:
GDC-0927 is a novel,non-steroidal, potent, orally bioavailable, selective estrogen receptor antagonist.
CAS:
1642297-01-5
Formula:
C28H28FNO4
Molecular Weight:
461.533
Purity:
0.98
SMILES:
CC1=C([C@@H](Oc2ccc(O)cc12)c1ccc(OCCN2CC(CF)C2)cc1)c1cccc(O)c1

References

1. MN Dickler, et al. Abstract PD5-10: A first-in-human phase I study to evaluate the oral selective estrogen receptor degrader (SERD), GDC-0927, in postmenopausal women with estrogen receptor positive (ER+) HER2-negative metastatic breast cancer (BC). AACR; Cancer Res 2018;78(4 Suppl):Abstract nr PD5-10.