TargetMol

Umbralisib R-enantiomer

Product Code:
 
TAR-T13140
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T13140-1mg1mg£258.00
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TAR-T13140-2mg2mg£348.00
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TAR-T13140-5mg5mg£539.00
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TAR-T13140-1mL1 mL * 10 mM (in DMSO)£734.00
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TAR-T13140-10mg10mg£741.00
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Quantity:
TAR-T13140-25mg25mg£1,091.00
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Quantity:
TAR-T13140-50mg50mg£1,428.00
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Quantity:
TAR-T13140-100mg100mg£1,910.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Umbralisib R-enantiomer (TGR-1202 R-enantiomer) is an inhibitor of PI3Kδ, which is the less active enantiomer of TGR-1202.
CAS:
1532533-69-9
Formula:
C31H24F3N5O3
Molecular Weight:
571.56
Pathway:
PI3K/Akt/mTOR signaling
Purity:
0.98
SMILES:
CC(C)Oc1ccc(cc1F)-c1nn([C@H](C)c2oc3ccc(F)cc3c(=O)c2-c2cccc(F)c2)c2ncnc(N)c12
Target:
PI3K

References

1. Michael Weiss, et al. Combination of anti-cd20 antibody and pi3 kinase selective inhibitor. WO2014071125A1.