TargetMol

URAT1 inhibitor 1

Product Code:
 
TAR-T13259
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T13259-5mg5mg£371.00
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Quantity:
TAR-T13259-50mg50mg£1,765.00
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Quantity:
TAR-T13259-100mg100mg£2,601.00
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This product comes from: United States.
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Further Information

Bioactivity:
URAT1 inhibitor 1 (1g) is an inhibitor of uric acid transporter 1 (URAT1) (IC50: 32 nM), has the potential to treat hyperuricemia associated with gout.
CAS:
2268720-62-1
Formula:
C19H15Br2N5O2S2
Molecular Weight:
569.29
Pathway:
Membrane transporter/Ion channel
Purity:
0.98
SMILES:
Brc1nnc(SCS(=O)(=O)Nc2cccnc2)n1Cc1ccc(Br)c2ccccc12
Target:
OAT

References

1. Wu JW, et al. Synthesis, biological evaluation and 3D-QSAR studies of 1,2,4-triazole-5-substituted carboxylic acid bioisosteres as uric acid transporter 1 (URAT1) inhibitors for the treatment of hyperuricemia associated with gout. Bioorg Med Chem Lett. 2019 Feb 1;29(3):383-388.