TargetMol

TR antagonist 1

Product Code:
 
TAR-T13435
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T13435-5mg5mg£437.00
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Quantity:
TAR-T13435-50mg50mg£1,765.00
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Quantity:
TAR-T13435-100mg100mg£2,697.00
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This product comes from: United States.
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Further Information

Bioactivity:
TR antagonist 1 is a high-affinity antagonist of thyroid hormone receptor (TR) (IC50s of 36 and 22 nM for TRα and TRβ, respectively).
CAS:
500794-88-7
Formula:
C25H23Br2NO4
Molecular Weight:
561.27
Purity:
0.98
SMILES:
CC(C)c1cc(Oc2c(Br)cc(CCC(O)=O)cc2Br)cc(C=Cc2ccncc2)c1O

References

1. Koehler K, et al. Thyroid receptor ligands. 6. A high affinity "direct antagonist" selective for the thyroid hormone receptor. J Med Chem. 2006 Nov 16;49(23):6635-7.