TargetMol

ACT-709478

Product Code:
 
TAR-T14120
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T14120-100mg100mgEnquire
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TAR-T14120-50mg50mgEnquire
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This product comes from: United States.
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Further Information

Bioactivity:
ACT-709478 is a potent, selective, orally active, and brain penetrating T-type calcium channel blocker. ACT-709478 is used in the research of generalized epilepsies[1].
CAS:
1838651-58-3
Formula:
C22H18F3N5O
Molecular Weight:
425.415
Purity:
0.98
SMILES:
FC(F)(F)C1(CC1)c1ccc(CC(=O)Nc2ccn(Cc3ccc(cn3)C#N)n2)cc1

References

1. Bezen?on O, et al. Discovery of a Potent, Selective T-type Calcium Channel Blocker as a Drug Candidate for the Treatment of Generalized Epilepsies. J Med Chem. 2017 Dec 14;60(23):9769-9789.